CP 55,244
Encyclopedia
CP 55,244 is a compound which is a cannabinoid receptor agonist. It has analgesic
effects and is used in scientific research. It is an extremely potent CB1 full agonist with a Ki
of 0.21nM, making it more potent than the commonly used full agonist HU-210
.
Analgesic
An analgesic is any member of the group of drugs used to relieve pain . The word analgesic derives from Greek an- and algos ....
effects and is used in scientific research. It is an extremely potent CB1 full agonist with a Ki
Dissociation constant
In chemistry, biochemistry, and pharmacology, a dissociation constant is a specific type of equilibrium constant that measures the propensity of a larger object to separate reversibly into smaller components, as when a complex falls apart into its component molecules, or when a salt splits up into...
of 0.21nM, making it more potent than the commonly used full agonist HU-210
HU-210
HU-210 is a synthetic cannabinoid that was first synthesized in 1988 from -Myrtenol by the group led by Professor Raphael Mechoulam at the Hebrew University. HU-210 is 100 to 800 times more potent than natural THC from cannabis and has an extended duration of action...
.