Bufuralol
Encyclopedia
Bufuralol is a potent beta-adrenoceptor antagonist with partial agonist
activity. It is metabolized by CYP2D6
.
Partial agonist
Partial agonists bind and activate a given receptor, but have only partial efficacy at the receptor relative to a full agonist...
activity. It is metabolized by CYP2D6
CYP2D6
Cytochrome P450 2D6 , a member of the cytochrome P450 mixed-function oxidase system, is one of the most important enzymes involved in the metabolism of xenobiotics in the body. Also, many substances are bioactivated by CYP2D6 to form their active compounds...
.